Biological study on novel coumarinyl 1,3,4-oxadiazoles

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منابع مشابه

Combined in Vitro and in Silico Studies for the Anticholinesterase Activity and Pharmacokinetics of Coumarinyl Thiazoles and Oxadiazoles

Citation: Ibrar A, Khan A, Ali M, Sarwar R, Mehsud S, Farooq U, Halimi SMA, Khan I and Al-Harrasi A (2018) Combined in Vitro and in Silico Studies for the Anticholinesterase Activity and Pharmacokinetics of Coumarinyl Thiazoles and Oxadiazoles. Front. Chem. 6:61. doi: 10.3389/fchem.2018.00061 Combined in Vitro and in Silico Studies for the Anticholinesterase Activity and Pharmacokinetics of Cou...

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A new and efficient method for the synthesis of novel 3-acetyl coumarins oxadiazoles derivatives with expected biological activity.

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Study on the synthesis of novel 5-substituted 2-[2-(pyridyl)ethenyl]-1,3,4-oxadiazoles and their acid–base interactions

ABSTRACT A series of novel 5-substituted 2-[2-(pyridyl)ethenyl]-1,3,4-oxadiazoles were efficiently synthesized by cyclocondensation of the appropriate 3-(pyridyl)acrylohydrazides with triethyl orthoesters in the presence of glacial acetic acid. The products were identified by means of spectroscopic methods and their pKA ionization constants were determined. The influence of substituents on the ...

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Synthesis and Characterization of New 2,5-disubstituted-1,3,4- oxadiazoles as Possible Biological Active Compounds

GABRIELA LAURA ALMAJAN1*, STEFANIA-FELICIA BARBUCEANU1, ILEANA FARCASANU2, CONSTANTIN DRAGHICI3 1 University of Medicine and Pharmacy, Faculty of Pharmacy, Organic Chemistry Department, 6 Traian Vuia Street, 020956 Bucharest, Romania 2 University of Bucharest, Faculty of Chemistry, Organic Chemistry, Biochemistry and Catalysis Department, 90-92 Sos. Panduri, 050663, Bucharest, Romania 3 Romania...

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ژورنال

عنوان ژورنال: TURKISH JOURNAL OF CHEMISTRY

سال: 2018

ISSN: 1300-0527,1303-6130

DOI: 10.3906/kim-1703-2